0001036050-00-001012 S-1 21 20000523 3 DIMENSIONAL PHARMACEUTICALS INC 0000914201 232716487 DE 1231 S-1 33 333-37606 641751 665 STOCKTON DRIVE SUITE 104 EXTON PA 19341 6104588959 665 STOCKTON DRIVE SUITE 104 EXTON PA 19341 S-1 1 000103605000001012-001-seq1-s-1.txt REGISTRATION STATEMENT EX-10.2 2 000103605000001012-002-seq2-ex-10-2.txt 3RD AMENDED STOCKHOLDERS AGREEMENT EX-10.3 3 000103605000001012-003-seq3-ex-10-3.txt SERIES B PREFERRED STOCK PURCHASE AGREEMENT EX-10.4 4 000103605000001012-004-seq4-ex-10-4.txt SERIES C PREFERRED STOCK PURCHASE AGREEMENT EX-10.6 5 000103605000001012-005-seq5-ex-10-6.txt WARRANT TO PURCHASE COMMON STOCK HEALTHCARE III EX-10.7 6 000103605000001012-006-seq6-ex-10-7.txt WARRANT TO PURCHASE COMMON STOCK TO HEALTHCARE IV EX-10.8 7 000103605000001012-007-seq7-ex-10-8.txt WARRANT TO PURCHASE COMMON STOCK TO RHO EX-10.9 8 000103605000001012-008-seq8-ex-10-9.txt WARRANT TO PURCHASE COMMON STOCK TO AETNA EX-10.10 9 000103605000001012-009-seq9-ex-10-10.txt WARRANT TO PURCHASE COMMON STOCK TO H. ROTHMAN EX-10.11 10 000103605000001012-010-seq10-ex-10-11.txt WARRANT TO PURCHASE COMMON STOCK TO ABINGWORTH BIO EX-10.12 11 000103605000001012-011-seq11-ex-10-12.txt WARRANT TO PURCHASE COMMON STOCK TO SENTRON MED EX-10.13 12 000103605000001012-012-seq12-ex-10-13.txt WARRANT TO PURCHASE COMMON STOCK TO BIOTECH GROWTH EX-10.15 13 000103605000001012-013-seq13-ex-10-15.txt SETTLEMENT AGMNT BTWN THE COMPANY & SCRIPTGEN EX-10.16 14 000103605000001012-014-seq14-ex-10-16.txt RESEARCH AGMNT BTWN THE COMPANY & BIOCRYST PHARM. EX-10.17 15 000103605000001012-015-seq15-ex-10-17.txt DISCOVERY & LEAD OPTI AGMNT BTWN COMPANY & BOEHRINGER EX-10.18 16 000103605000001012-016-seq16-ex-10-18.txt RESEARCH & LICENSE AGMNT BTWN COMPANY & HOECHST EX-10.19 17 000103605000001012-017-seq17-ex-10-19.txt RESEARCH & LICENSE AGMNT BTWN COMPANY & DUPONT EX-10.22 18 000103605000001012-018-seq18-ex-10-22.txt RESEARCH & LICENSE AGMNT BTWN COMPANY & HESKA EX-21.1 19 000103605000001012-019-seq19-ex-21-1.txt SUBSIDIARIES OF THE REGISTRANT EX-23.1 20 000103605000001012-020-seq20-ex-23-1.txt CONSENT OF RICHARD A. EISNER & CO. L.L.P. EX-27.1 21 000103605000001012-021-seq21-ex-27-1.txt FINANCIAL DATA SCHEDULE